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S.No PRODUCT CAS NO STRUCTURE THERAPEUTIC APPLICATION
1 ACEBUTOLOL 37517-30-9 Antiarrhythmics (Beta blockers) (Group II); Beta-adrenergic blocking agents :cardioselective beta blockers;Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor Agonists
2ACETAZOLAMIDE 59-66-5 Diuretics (Carbonic anhydrase inhibitors)
3 ADENOSINE 58-61-7 Adenosine receptor modulator agonists; Antiarrhythmics (Group V)
4 ALFUZOSIN 81403-80-7 Alpha-adrenoceptor blockers (alpha-blockers)
5 ALISKIREN 173334-57-1 Renin inhibitors
6 ALPROSTADIL 745-65-3 Direct-acting Vasodilators
7 AMBRISENTAN 177036-94-1 Endothelin receptor antagonists
8 AMILORIDE HYDROCHLORIDE2016-88-8 Diuretics (Potassium-sparing diuretics)
9 AMIODARONE 1951-25-3 Antiarrhythmics: Potassium-channel blockers (Group III)
10 AMLODIPINE88150-42-9 Antiarrhythmics: Calcium-channel blockers (Group IV)
11 APADENOSON 250386-15-3 Selective A2a adenosine receptor agonist
12 ATENOLOL29122-68-7 Cardioselective beta blockers; Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
13 ATROPINE 51-55-8 Muscarinic receptor antagonists; Anticholinergic chronotropic agents ( also known as muscarinic antagonists or parasympatholytic)Positive chronotropes
14 ATORVASTATIN134523-00-5 HMG-CoA reductase inhibitors
15 AZILSARTAN147403-03-0 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
16 BENAZEPRIL 86541-75-5 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
17 BETAXOLOL 63659-18-7 Beta-adrenergic blocking agents (cardioselective beta blockers) ; Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
18 BINODENOSON144348-08-3 Adenosine receptor modulator agonist
19 BISOPROLOL66722-44-9 Beta-adrenergic blocking agents (cardioselective beta blockers); Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
20 BOSENTAN147536-97-8 Endothelin receptor antagonists
21 BRINZOLAMIDE138890-62-7 Diuretics (Carbonic anhydrase inhibitors)
22 BUFALIN465-21-4 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
23 BUMETANIDE 28395-03-1 Diuretics (loop)
24 CANAGLIFLOZIN842133-18-0 Sodium-glucose co-transporter 2 (SGLT-2) inhibitors
25 CANDESARTAN 139481-59-7 Angiotensin receptor blocker (ARBs or angiotensin II inhibitor)
26 CAPADENOSON 544417-40-5 Selective adenosine A1‐receptor agonist
27 CAPTOPRIL62571-86-2 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
28 CARVEDILOL72956-09-3 Non-selective β-adrenergic receptor antagonist (β1, β2) and an α-adrenergic receptor antagonist (α1)
29 CHLORISONDAMINE7701-62-4 Ganglionic blockers
30 CHLORTHALIDONE 77-36-1 Diuretics (thiazide)
31 CILOSTAZOL 73963-72-1 Peripheral vasodilators
32 CINOBUFAGIN470-37-1 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
33 CLONIDINE4205-90-7 Centrally acting antiadrenergic agents (sympatholytic)
34 CLOPIDOGREL 113665-84-2 Cardiovascular agent
35 CONIVAPTAN 210101-16-9 Vasopressin antagonists
36 CROMAKALIM94470-67-4 Potassium-channel openers
37 DABIGATRAN 211915-06-9 Fibrinolytic (thrombolytic)
38 DAPAGLIFLOZIN461432-26-8 Sodium-glucose co-transporter 2 (SGLT-2) inhibitors
39 DENOPAMINE 71771-90-9 Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
40 DIAZOXIDE 364-98-7 Potassium-channel openers
41 DICLOFENAMIDE 120-97-8 Diuretics (Carbonic anhydrase inhibitors)
42 DILTIAZEM 42399-41-7 Antiarrhythmics: Calcium-channel blockers (Group IV)
43 DISOPYRAMIDE 3737-09-5 Antiarrhythmics: Sodium-channel blockers (Group 1); (late sodium currents)
44 DOBUTAMINE 34368-04-2 Sympathomimetics; Vasopressors; Inotropic agents; Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor; Catecholamines
45 DOFETILIDE 115256-11-6 Antiarrhythmics: Potassium-channel blockers (Group III)
46 DORZOLAMIDE 120279-96-1 Diuretics (Carbonic anhydrase inhibitors)
47 DOXAZOSIN 74191-85-8 Alpha-adrenoceptor blockers (alpha-blockers)
48 DRONEDARONE 141626-36-0 Antiarrhythmics: Potassium-channel blockers (Group III)
49 EMPAGLIFLOZIN 864070-44-0 Sodium-glucose co-transporter 2 (SGLT-2) inhibitors
50 ENALAPRIL 75847-73-3 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
51 ENCAINIDE 66778-36-7 Sodium-channel blocker (late sodium currents)
52 EPHEDRINE 299-42-3 Vasopressors
53 EPINEPHRINE 51-43-4 Vasopressors; Sympathomimetics; Anticholinergic chronotropic agents ( also known as muscarinic antagonists or parasympatholytic) Positive chronotropes; Catecholamines
54 EPLERENONE 107724-20-9 Aldosterone receptor antagonists (ARAs) (also called an antimineralocorticoid, MCRA, and sometimes MRA); Diuretics (potassium-sparing)
55 EPROSARTAN 133040-01-4 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
56 ERTUGLIFLOZIN 1210344-57-2 Sodium-glucose co-transporter 2 (SGLT-2) inhibitors
57 ESMOLOL 81147-92-4 Beta-adrenergic blocking agents (cardioselective beta blockers); Antiarrhythmics (Beta blockers) (Group II)
58 ETHACRYNIC ACID 58-54-8 Diuretic agent (loop)
59 ETHANOLAMINE OLEATE 2272-11-9 Sclerosing agents
60 ETHOXZOLAMIDE 452-35-7 Diuretics (Carbonic anhydrase inhibitors)
61 FINERENONE 1050477-31-0 Funny current blockers; Aldosterone receptor antagonists (ARAs) (also called an antimineralocorticoid, MCRA, and sometimes MRA);
62 FLECAINIDE 54143-55-4 Sodium-channel blocker (late sodium currents)
63 FLUPIRTINE 56995-20-1 Potassium-channel openers
64 FLUVASTATIN 93957-54-1 HMG-CoA reductase inhibitors
65 FOSINOPRIL 98048-97-6 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
66 FUROSEMIDE 54-31-9 Diuretic agent (loop)
67 GABAPENTIN 60142-96-3 HCN channel Blockers
68 GUANABENZ 5051-62-7 Centrally acting antiadrenergic agents (sympatholytic)
69 GUANFACINE 29110-47-2 Centrally acting antiadrenergic agents (sympatholytic)
70 HEXAMETHONIUM 60-26-4 Ganglionic blockers
71 HYDRALAZINE 86-54-4 Nitrodilators; Direct-acting Vasodilators
72 HYDROCHLOROTHIAZIDE 58-93-5 Diuretics (thiazide)
73 IBUTILIDE 122647-31-8 Antiarrhythmics: Potassium-channel blockers (Group III)
74 INDAPAMIDE 26807-65-8 Diuretics (thiazide)
75 IRBESARTAN 138402-11-6 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
76 ISOPROTERENOL 7683-59-2 Vasopressors; Sympathomimetics; Anticholinergic chronotropic agents ( also known as muscarinic antagonists or parasympatholytic) Positive chronotropes; Catecholamines
77 ISORDIL 87-33-2 Nitrodilators
78 ISOSORBIDE MONONITRATE 16051-77-7 Antianginal agents
79 ISOTRATE 652-67-5 Nitrodilators
80 IVABRADINE 155974-00-8 HCN channel blockers; Funny current blockers
81 LABETALOL 36894-69-6 Beta-adrenergic blocking agents
82 LIDOCAINE 137-58-6 Antiarrhythmics: Sodium-channel blockers (Group 1) (late sodium currents);
83 (S)-LISINOPRIL DIHYDRATE 83915-83-7 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
84 LOFEXIDINE 31036-80-3 Centrally acting antiadrenergic agents (sympatholytic)
85 LOSARTAN 114798-26-4 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
86 LOVASTATIN 75330-75-5 HMG-CoA reductase inhibitors
87 MACITENTAN 441798-33-0 Endothelin receptor antagonists
88 MAVACAMTEN 1642288-47-8 Cardiovascular agent
89 MEXILETINE 31828-71-4 Antiarrhythmics: Sodium-channel blockers (Group 1); (late sodium currents)
90 METOPROLOL51384-51-1 Cardioselective beta blockers; Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor; Funny current blockers
91 METHAZOLAMIDE 554-57-4 Diuretics (Carbonic anhydrase inhibitors)
92 METOLAZONE17560-51-9 Diuretics (thiazide)
93 METHYCLOTHIAZIDE 135-07-9 Diuretics (thiazide)
94 MECAMYLAMINE 6147-18-8 Ganglionic blockers
95 MILRINONE 78415-72-2 Anticholinergic chronotropic agents ( also known as muscarinic antagonists or parasympatholytic)Positive chronotropes; Inotropic agents
96 MINOXIDIL 38304-91-5 Potassium-channel openers; Direct-acting Vasodilators
97 MOEXIPRIL 103775-10-6 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
98 MORICIZINE 31883-05-3 Antiarrhythmics: Sodium-channel blockers (Group 1); (late sodium currents)
99 MOXISYLYTE 54-32-0 Peripheral vasodilators
100 NADOLOL 42200-33-9 Beta-adrenergic blocking agents
101 NAFTIDROFURYL 31329-57-4 Peripheral vasodilators
102 NEBIVOLOL 118457-14-0 Cardioselective beta blockers; Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
103 NELADENOSON BIALANATE 1239309-58-0 Adenosine receptor modulator agonists
104 NERIIFOLIN 466-07-9 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
105 NICORANDIL 65141-46-0 Potassium-channel openers
106 NIFEDIPINE 21829-25-4 Peripheral vasodilators
107 NITROGLYCERIN 55-63-0 Antianginal agents; Direct-acting Vasodilators
108 NORADRENALINE 51-41-2 Beta-adrenoceptor agonists
109 OLEANDRIN 465-16-7 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
110 OLMESARTAN MEDOXOMIL 144689-63-4 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
111 OMECAMTIV MECARBIL 873697-71-3 Funny current blockers
112 ORVATEN 42794-76-3 Cardiovascular agent
113 OUABAIN 630-60-4 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
114 PEIMISINE 19773-24-1 Muscarinic receptor antagonists
115 PEMPIDINE 79-55-0 Ganglionic blockers
116 PENBUTOLOL 38363-40-5 Beta-adrenergic blocking agents
117 PENTOLINIUM 144-44-5 Ganglionic blockers
118 PENTOXIFYLLINE 6493-05-6 Peripheral vasodilators
119 PERINDOPRIL 82834-16-0 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
120 PINACIDIL 60560-33-0 Nonselective beta blocker
121 PINDOLOL 13523-86-9 Beta-adrenergic blocking agents
122 PITAVASTATIN 147511-69-1 HMG-CoA reductase inhibitors
123 PHENYLEPHRINE 59-42-7 Vasopressors
124 PHENYTOIN 57-41-0 Antiarrhythmics: Sodium-channel blockers (Group 1) (late sodium currents)
125 PHLORIZIN 60-81-1 Cardiac glycosides (Na+-K+- ATPase pump inhibitors)
126 PRAVASTATIN 81093-37-0 HMG-CoA reductase inhibitors
127 PRAZOSIN 19216-56-9 Alpha-adrenoceptor blockers (alpha-blockers)
128 PROCAINAMIDE 51-06-9 Antiarrhythmics: Sodium-channel blockers (Group 1) (late sodium currents)
129 PROPAFENONE 54063-53-5 Antiarrhythmics: Sodium-channel blockers (Group 1) (late sodium currents)
130 PROPRANOLOL 525-66-6 Antiarrhythmics (Beta blockers) (Group II); Beta-adrenergic blocking agents
131 QUINAPRIL 85441-61-8 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
132 QUINIDINE 56-54-2 Antiarrhythmics: Sodium-channel blockers (Group 1) (late sodium currents)
133 RAMIPRIL 87333-19-5 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
134 RANOLAZINE 95635-55-5 Antianginal agents
135 REGADENOSON 313348-27-5 Adenosine receptor modulator agonists
136 REMIKIREN 126222-34-2 Renin inhibitors
137 RETIGABINE 150812-12-7 Potassium-channel openers
138 RIOCIGUAT 625115-55-1 Direct-acting vasodilators
139 ROSUVASTATIN 287714-41-4 HMG-CoA reductase inhibitors
140 SACUBITRIL 149709-62-6 Neprilysin inhibitors (ARNI)
141 SARPOGRELATE 125926-17-2 Muscarinic receptor antagonists
142 SILDENAFIL 139755-83-2 Phosphodiesterase inhibitors
143 SILODOSIN 160970-54-7 Alpha adrenoreceptor antagonists (Selective α1-adrenergic receptor antagonists)
144 SIMVASTATIN 79902-63-9 HMG-CoA reductase inhibitors
145 SITAXSENTAN 184036-34-8 Endothelin receptor antagonists
146 SODIUM TETRADECYL SULFATE 139-88-8 Sclerosing agents
147 SOTALOL 3930-20-9 Antiarrhythmics: Potassium-channel blockers (Group III); Beta-adrenergic blocking agents
148 SPIRONOLACTONE 52-01-7 Aldosterone receptor antagonists (ARAs) (also called an antimineralocorticoid, MCRA, and sometimes MRA); Potassium-sparing diuretics
149 TADANAFIL 171596-29-5 Phosphodiesterase inhibitors
150 TAMSULOSIN 106133-20-4 Alpha adrenoreceptor antagonists(Selective α1-adrenergic receptor antagonists)
151 TELMISARTAN 144701-48-4 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors)
152 TERAZOSIN 63590-64-7 Alpha-adrenoceptor blockers (alpha-blockers)
153 THEOPHYLLINE 58-55-9 Anticholinergic chronotropic agents ( also known as muscarinic antagonists or parasympatholytic) Positive chronotropes
154 TIMOLOL 26839-75-8 Beta-adrenergic blocking agents
155 TOCAINIDE 41708-72-9 Antiarrhythmics: Sodium-channel blockers (Group 1), (late sodium currents)
156 TOLVAPTAN 150683-30-0 Vasopressin antagonists
157 TORSEMIDE 56211-40-6 Diuretics (loop)
158 TRANDOLAPRIL 87679-37-6 Angiotensin-converting enzyme inhibitors (ACE inhibitors)
159 TRIAMTERENE 396-01-0 Diuretics (Potassium-sparing)
160 TRIMETAPHAN CAMSILATE 68-91-7 Ganglionic blockers
161 VALSARTAN 137862-53-4 Angiotensin receptor blockers (also called ARBs or angiotensin II inhibitors); Neprilysin inhibitors (ARNI)
162 VARDENAFIL 224785-90-4 Phosphodiesterase inhibitors
163 VERAPAMIL 52-53-9 Antiarrhythmics; Calcium-channel blockers (Group IV)
164 VERICIGUAT 1350653-20-1 Direct-acting vasodilators; Funny current blocker
165 VORTIOXETINE 508233-74-7 Beta-adrenoceptor antagonists (as beta blockers)
166 XAMOTEROL 81801-12-9 Beta-adrenoceptor agonists (beta1-agonists) also known as ADRB1, is a beta-adrenergic receptor
167 YM758 312752-86-6 Funny current blockers
168 ZD-7288 133059-99-1 HCN channel blockers
169 ZONISAMIDE 68291-97-4 Diuretics (Carbonic anhydrase inhibitors)

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Disclaimer: Building blocks, key intermediates, and impurities associated with the above products protected by valid patents are not offered for sale in countries where the sale of such products constitutes patent infringement. Availability may be restricted to certain markets or countries.

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